Growth Hormone Secretagogues

Ipamorelin

Also known as: NNC 26-0161

Selective ghrelin-mimetic that triggers GH release without raising cortisol, ACTH, or prolactin. Often stacked with a GHRH analog like CJC-1295. Never administer IV (documented fatality risk), SubQ only.

Pharmacokinetics

Half-life
2 hours
Time to peak
15 min
Bioavailability
100%
Onset
15 min
Dosing interval
24h

Administration

Primary routes
SubQ
Category
Growth Hormone Secretagogues

Safety Flags

  • High immunogenicity
  • Contraindicated in cancer history

Storage

  • · Requires refrigeration (2–8°C)
  • · Temperature sensitive — minimise room-temp exposure